Synthesis and microbiological activity of some 2H-1,4-benzothiazin-3-one derivatives.
dc.contributor.author | Guarda, Vera Lúcia de Miranda | |
dc.contributor.author | Perrissin, Monique | |
dc.contributor.author | Thomasson, François | |
dc.contributor.author | Ximenes, Eulália Camelo Pessoa de Azevedo | |
dc.contributor.author | Galdino, Suely Lins | |
dc.contributor.author | Pitta, Ivan da Rocha | |
dc.contributor.author | Luu-Duc, Cuong | |
dc.date.accessioned | 2017-04-26T15:41:37Z | |
dc.date.available | 2017-04-26T15:41:37Z | |
dc.date.issued | 2000 | |
dc.description.abstract | The synthesis and physicochemical properties of 4-butyl-2H-benzo[1,4]thiazin-3-one derivatives are described. These new compounds were synthesised by alkylation in 4-N position and acylation and/or alkylation of 6-NH2 by phase transfer catalysis. Acid hydrolysis of 6-alkylacylamino group yielded 6-alkylamino-4-butyl-2H-benzo[1,4]thiazin-3-ones. The antimicrobial in vitro activity was determined on five compounds. | pt_BR |
dc.identifier.citation | GUARDA, V. L. de M. et al. Synthesis and microbiological activity of some 2H-1,4-benzothiazin-3-one derivatives. Heterocyclic Communications, v. 06, n.01, p. 35-40, 2000. Disponível em: <https://www.degruyter.com/view/j/hc.2000.6.1/hc.2000.6.1.49/hc.2000.6.1.49.xml>. Acesso em: 20 jan. 2017. | pt_BR |
dc.identifier.doi | https://doi.org/10.1515/HC.2000.6.1.49 | |
dc.identifier.issn | 2191-0197 | |
dc.identifier.uri | http://www.repositorio.ufop.br/handle/123456789/7636 | |
dc.identifier.uri2 | https://www.degruyter.com/view/j/hc.2000.6.1/hc.2000.6.1.49/hc.2000.6.1.49.xml | pt_BR |
dc.language.iso | en_US | pt_BR |
dc.rights | restrito | pt_BR |
dc.subject | Benzothiazines | pt_BR |
dc.subject | Antimicrobial activity | pt_BR |
dc.title | Synthesis and microbiological activity of some 2H-1,4-benzothiazin-3-one derivatives. | pt_BR |
dc.type | Artigo publicado em periodico | pt_BR |